Wednesday, July 8, 2026

Drug profile · INN

atenolol

atenolol (APX-ATENOLOL) is a beta-1 adrenergic receptor antagonist. Associated with Alphapharm Pty Ltd. Route of administration: injection. Current US regulatory status: approved.

FDA: approved TGA: approved
US status approved
Patents linked 20
Pipeline programs 2
News articles 0
Drug details — atenolol
US status
approved
Class
Route
INJECTION
Patents
20
Programs
2
Data quality
0.89

Quick answer

atenolol (APX-ATENOLOL) is a beta-1 adrenergic receptor antagonist. Associated with Alphapharm Pty Ltd. Route of administration: injection. Current US regulatory status: approved.

Key facts

INN atenolol
Brand APX-ATENOLOL
Mechanism Beta-1 adrenergic receptor antagonist
Target Beta-1 adrenergic receptor
Route INJECTION
Formulation INJECTABLE

Mechanism of action

Beta-1 adrenergic receptor antagonist

Primary target: Beta-1 adrenergic receptor

Approval history

Authority Status Date
FDA approved
TGA approved

Pipeline programs

  1. Atenolol Approved · Cardiff Oncology · Marfan Syndrome
  2. BA-SCAD Approved · Cardiol Therapeutics · Spontaneous Coronary Artery Dissection.

Related & competitor drugs

  1. acebutolol hydrochloride Beta-1 adrenergic receptor antagonist
  2. bisoprolol fumarate Beta-1 adrenergic receptor antagonist
  3. dobutamine hydrochloride Beta-1 adrenergic receptor agonist
  4. dopamine hydrochloride Cardiovascular system (C01)
  5. esmolol hydrochloride Beta-2 adrenergic receptor antagonist
  6. metoprolol succinate Beta-1 adrenergic receptor antagonist
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Frequently asked questions

What is atenolol?

atenolol (APX-ATENOLOL) is a beta-1 adrenergic receptor antagonist. Associated with Alphapharm Pty Ltd. Route of administration: injection. Current US regulatory status: approved.

What is the brand name for atenolol?

APX-ATENOLOL is a marketed brand name for atenolol. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of atenolol?

atenolol has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.