Wednesday, June 10, 2026

pharma Β· Carcinoma, Non-small-cell Lung Β· Type 2 Diabetes Mellitus Β· LGND

LIGAND PHARMACEUTICALS

LIGAND PHARMACEUTICALS drug portfolio β€” 25 indexed compounds with therapeutic class and molecular targets from public FDA and regional approval metadata.

555 Heritage Dr, Suite 200, Jupiter, Florida 33458, US HQ
1987 Founded
130 Employees
Public company Type
LGND Β· NYSE Ticker
Company details
Status
Public
HQ
555 Heritage Dr, Suite 200, Jupiter, Florida 33458, US
Founded
1987
Employees
130
Programs
34
Drugs
25
Patents
133
Intelligence Β· Drug Pipeline

LIGAND PHARMACEUTICALS pipeline

Portfolio lens on 25 drugs and development assets β€” regulatory status, targets, and deep links to NovaPharmaNews drug profiles.

LIGAND PHARMACEUTICALS drug portfolio β€” 25 indexed compounds with therapeutic class and molecular targets from public FDA and regional approval metadata.

Drug portfolio

25 compounds
  1. alitretinoin

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Retinoid receptor.

    Target
    Retinoid receptor
    Mechanism
    Retinoid receptor agonist
  2. bexarotene

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Retinoid X receptor.

    Target
    Retinoid X receptor
    Mechanism
    Retinoid X receptor agonist
  3. budesonide

    Alimentary tract and metabolism (A07)

    US regulatory status: approved. Molecular target: Glucocorticoid receptor.

    Target
    Glucocorticoid receptor
    Mechanism
    Glucocorticoid receptor agonist
  4. US regulatory status: approved. Molecular target: Sodium channel alpha subunit.

    Target
    Sodium channel alpha subunit
    Mechanism
    Sodium channel alpha subunit blocker
  5. US regulatory status: approved. Molecular target: Solute carrier family 12 member 3.

    Target
    Solute carrier family 12 member 3
    Mechanism
    Thiazide-sensitive sodium-chloride cotransporter inhibitor
  6. US regulatory status: approved. Molecular target: Elongation factor 2.

    Target
    Elongation factor 2
    Mechanism
    Interleukin-2 receptor binding agent
  7. US regulatory status: approved. Molecular target: Glucocorticoid receptor.

    Target
    Glucocorticoid receptor
    Mechanism
    Glucocorticoid receptor agonist
  8. erlotinib

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in LIGAND PHARMACEUTICALS's portfolio. Mechanism: Epidermal growth factor receptor erbB1 inhibitor.

    Mechanism
    Epidermal growth factor receptor erbB1 inhibitor
  9. US regulatory status: approved. Molecular target: Epidermal growth factor receptor.

    Target
    Epidermal growth factor receptor
    Mechanism
    Epidermal growth factor receptor erbB1 inhibitor
  10. US regulatory status: approved. Molecular target: Solute carrier family 12 member 3.

    Target
    Solute carrier family 12 member 3
    Mechanism
    Thiazide-sensitive sodium-chloride cotransporter inhibitor
  11. Development asset linked to LIGAND PHARMACEUTICALS in public FDA and regional records.

  12. US regulatory status: approved. Mechanism: Diagnostic agent.

    Mechanism
    Diagnostic agent
  13. irbesartan

    Cardiovascular system (C09)

    US regulatory status: approved. Molecular target: Type-1 angiotensin II receptor.

    Target
    Type-1 angiotensin II receptor
    Mechanism
    Type-1 angiotensin II receptor antagonist
  14. lasofoxifene

    Genito-urinary system and sex hormones (G03)

    Genito-urinary system and sex hormones (G03) compound in LIGAND PHARMACEUTICALS's portfolio. Molecular target: Estrogen receptor.

    Target
    Estrogen receptor
    Mechanism
    Estrogen receptor modulator
  15. Development asset linked to LIGAND PHARMACEUTICALS in public FDA and regional records.

  16. Development asset linked to LIGAND PHARMACEUTICALS in public FDA and regional records.

  17. Development asset linked to LIGAND PHARMACEUTICALS in public FDA and regional records.

  18. US regulatory status: approved. Molecular target: Angiotensin-converting enzyme.

    Target
    Angiotensin-converting enzyme
    Mechanism
    Angiotensin-converting enzyme inhibitor
  19. Development asset linked to LIGAND PHARMACEUTICALS in public FDA and regional records.

  20. Development asset linked to LIGAND PHARMACEUTICALS in public FDA and regional records.

  21. Development asset linked to LIGAND PHARMACEUTICALS in public FDA and regional records.

  22. US regulatory status: approved. Molecular target: Retinoic acid receptor.

    Target
    Retinoic acid receptor
    Mechanism
    Retinoic acid receptor agonist