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Eli Lilly and

Eli Lilly and drug portfolio — 42 indexed compounds with therapeutic class and molecular targets from public FDA and regional approval metadata.

Lilly Corporate Center, Indianapolis, Indiana 46285, US HQ
55,860 Employees
NMPA registrant Type
Company details
Status
Public
HQ
Lilly Corporate Center, Indianapolis, Indiana 46285, US
Employees
55,860
Programs
62
Drugs
42
Patents
0
Intelligence · Drug Pipeline

Eli Lilly and pipeline

Portfolio lens on 42 drugs and development assets — regulatory status, targets, and deep links to NovaPharmaNews drug profiles.

Eli Lilly and drug portfolio — 42 indexed compounds with therapeutic class and molecular targets from public FDA and regional approval metadata.

Drug portfolio

42 compounds
  1. abacavir

    Antiinfectives for systemic use (J05)

    US regulatory status: approved.

  2. abemaciclib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Cyclin-dependent kinase 4.

    Target
    Cyclin-dependent kinase 4
    Mechanism
    Cyclin-dependent kinase 6 inhibitor
  3. US regulatory status: approved. Molecular target: GABA-A receptor; anion channel.

    Target
    GABA-A receptor; anion channel
    Mechanism
    GABA-A receptor; anion channel positive modulator
  4. Development asset linked to Eli Lilly and in public FDA and regional records.

  5. Various (V09) compound in Eli Lilly and's portfolio. Mechanism: Diagnostic agent.

    Mechanism
    Diagnostic agent
  6. baricitinib

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Molecular target: Tyrosine-protein kinase JAK1.

    Target
    Tyrosine-protein kinase JAK1
    Mechanism
    Tyrosine-protein kinase JAK2 inhibitor
  7. Development asset linked to Eli Lilly and in public FDA and regional records.

  8. clopidogrel

    Blood and blood forming organs (B01)

    Blood and blood forming organs (B01) compound in Eli Lilly and's portfolio. Mechanism: Purinergic receptor P2Y12 antagonist.

    Mechanism
    Purinergic receptor P2Y12 antagonist
  9. donanemab

    Nervous system (N06)

    Nervous system (N06) compound in Eli Lilly and's portfolio. Molecular target: Amyloid-beta precursor protein.

    Target
    Amyloid-beta precursor protein
    Mechanism
    Beta amyloid A4 protein disrupting agent
  10. drotrecogin alfa (activated)

    Blood and blood forming organs (B01)

    Blood and blood forming organs (B01) compound in Eli Lilly and's portfolio. Molecular target: Coagulation factor V.

    Target
    Coagulation factor V
    Mechanism
    Coagulation factor V inhibitor
  11. duloxetine

    Nervous system (N06)

    Nervous system (N06) compound in Eli Lilly and's portfolio. Mechanism: Serotonin transporter inhibitor.

    Mechanism
    Serotonin transporter inhibitor
  12. US regulatory status: approved. Molecular target: Sodium-dependent noradrenaline transporter.

    Target
    Sodium-dependent noradrenaline transporter
    Mechanism
    Norepinephrine transporter inhibitor
  13. Development asset linked to Eli Lilly and in public FDA and regional records.

  14. US regulatory status: approved. Molecular target: Peroxisome proliferator-activated receptor alpha.

    Target
    Peroxisome proliferator-activated receptor alpha
    Mechanism
    Peroxisome proliferator-activated receptor alpha agonist
  15. Development asset linked to Eli Lilly and in public FDA and regional records. Molecular target: Insulin receptor.

    Target
    Insulin receptor
    Mechanism
    Insulin receptor agonist
  16. Development asset linked to Eli Lilly and in public FDA and regional records.

  17. Development asset linked to Eli Lilly and in public FDA and regional records.

  18. Development asset linked to Eli Lilly and in public FDA and regional records. Molecular target: Insulin receptor.

    Target
    Insulin receptor
    Mechanism
    Insulin receptor agonist
  19. insulin glargine

    Alimentary tract and metabolism (A10)

    US regulatory status: approved. Molecular target: Insulin receptor.

    Target
    Insulin receptor
    Mechanism
    Insulin receptor agonist
  20. insulin lispro

    Alimentary tract and metabolism (A10)

    US regulatory status: approved. Molecular target: Insulin receptor.

    Target
    Insulin receptor
    Mechanism
    Insulin receptor agonist
  21. Development asset linked to Eli Lilly and in public FDA and regional records.

  22. lebrikizumab

    Dermatologicals (D11)

    Dermatologicals (D11) compound in Eli Lilly and's portfolio. Molecular target: Interleukin-13.

    Target
    Interleukin-13
    Mechanism
    Interleukin-13 inhibitor
  23. Development asset linked to Eli Lilly and in public FDA and regional records.

  24. Development asset linked to Eli Lilly and in public FDA and regional records.

  25. Development asset linked to Eli Lilly and in public FDA and regional records.

  26. mirikizumab

    Antineoplastic and immunomodulating agents (L04)

    Antineoplastic and immunomodulating agents (L04) compound in Eli Lilly and's portfolio. Molecular target: Interleukin-23.

    Target
    Interleukin-23
    Mechanism
    Interleukin-23 inhibitor
  27. necitumumab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Epidermal growth factor receptor.

    Target
    Epidermal growth factor receptor
    Mechanism
    Epidermal growth factor receptor erbB1 inhibitor
  28. olaratumab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Platelet-derived growth factor receptor alpha.

    Target
    Platelet-derived growth factor receptor alpha
    Mechanism
    Platelet-derived growth factor receptor alpha antagonist
  29. Development asset linked to Eli Lilly and in public FDA and regional records.

  30. US regulatory status: approved. Molecular target: Dihydrofolate reductase.

    Target
    Dihydrofolate reductase
    Mechanism
    Thymidylate synthase inhibitor
  31. US regulatory status: approved. Molecular target: Dihydrofolate reductase.

    Target
    Dihydrofolate reductase
    Mechanism
    Thymidylate synthase inhibitor
  32. Development asset linked to Eli Lilly and in public FDA and regional records.

  33. Development asset linked to Eli Lilly and in public FDA and regional records.

  34. propranolol

    Cardiovascular system (C07)

    Cardiovascular system (C07) compound in Eli Lilly and's portfolio. Mechanism: Beta-1 adrenergic receptor antagonist.

    Mechanism
    Beta-1 adrenergic receptor antagonist
  35. ramucirumab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Vascular endothelial growth factor receptor 2.

    Target
    Vascular endothelial growth factor receptor 2
    Mechanism
    Vascular endothelial growth factor receptor 2 inhibitor
  36. selpercatinib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Coiled-coil domain-containing protein 6/Tyrosine-protein kinase receptor RET.

    Target
    Coiled-coil domain-containing protein 6/Tyrosine-protein kinase receptor RET
    Mechanism
    Tyrosine-protein kinase receptor RET inhibitor
  37. tadalafil

    Genito-urinary system and sex hormones (G04)

    US regulatory status: approved. Molecular target: cGMP-specific 3',5'-cyclic phosphodiesterase.

    Target
    cGMP-specific 3',5'-cyclic phosphodiesterase
    Mechanism
    Phosphodiesterase 5A inhibitor
  38. teriparatide

    Systemic hormonal preparations (H05)

    US regulatory status: approved. Molecular target: Parathyroid hormone/parathyroid hormone-related peptide receptor.

    Target
    Parathyroid hormone/parathyroid hormone-related peptide receptor
    Mechanism
    Parathyroid hormone receptor agonist
  39. testosterone

    Genito-urinary system and sex hormones (G03)

    US regulatory status: approved. Molecular target: Androgen receptor.

    Target
    Androgen receptor
    Mechanism
    Androgen Receptor agonist
  40. tirzepatide

    Alimentary tract and metabolism (A10)

    US regulatory status: approved. Molecular target: Gastric inhibitory polypeptide receptor.

    Target
    Gastric inhibitory polypeptide receptor
    Mechanism
    Glucagon-like peptide 1 receptor agonist