Wednesday, June 10, 2026

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Lxo Ireland Designated

Lxo Ireland Designated drug portfolio β€” 61 indexed compounds with therapeutic class and molecular targets from public FDA and regional approval metadata.

CARLSBAD, CA, IE HQ
Public company Type
DSGN Β· NYSE Ticker
Company details
Intelligence Β· Drug Pipeline

Lxo Ireland Designated pipeline

Portfolio lens on 61 drugs and development assets β€” regulatory status, targets, and deep links to NovaPharmaNews drug profiles.

Lxo Ireland Designated drug portfolio β€” 61 indexed compounds with therapeutic class and molecular targets from public FDA and regional approval metadata.

Drug portfolio

61 compounds
  1. abiraterone

    Antineoplastic and immunomodulating agents (L02)

    Antineoplastic and immunomodulating agents (L02) compound in Lxo Ireland Designated's portfolio. Molecular target: Androgen receptor.

    Target
    Androgen receptor
    Mechanism
    Steroid 5-alpha-reductase inhibitor
  2. Development asset linked to Lxo Ireland Designated in public FDA and regional records.

  3. alectinib

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Lxo Ireland Designated's portfolio. Mechanism: EML4-ALK.

    Mechanism
    EML4-ALK
  4. aliskiren

    Cardiovascular system (C09)

    Cardiovascular system (C09) compound in Lxo Ireland Designated's portfolio. Mechanism: Renin inhibitor.

    Mechanism
    Renin inhibitor
  5. Development asset linked to Lxo Ireland Designated in public FDA and regional records.

  6. Development asset linked to Lxo Ireland Designated in public FDA and regional records.

  7. Various (V09) compound in Lxo Ireland Designated's portfolio. Mechanism: Diagnostic agent.

    Mechanism
    Diagnostic agent
  8. Development asset linked to Lxo Ireland Designated in public FDA and regional records.

  9. Development asset linked to Lxo Ireland Designated in public FDA and regional records.

  10. atropine sulfate

    Sensory organs (S01)

    US regulatory status: approved. Molecular target: Muscarinic acetylcholine receptor M1.

    Target
    Muscarinic acetylcholine receptor M1
    Mechanism
    Muscarinic acetylcholine receptor M3 antagonist
  11. Development asset linked to Lxo Ireland Designated in public FDA and regional records.

  12. US regulatory status: approved. Mechanism: Unknown.

    Mechanism
    Unknown
  13. bupivacaine

    Nervous system (N01)

    US regulatory status: approved. Molecular target: Sodium channel protein type 4 subunit alpha.

    Target
    Sodium channel protein type 4 subunit alpha
    Mechanism
    Sodium channel protein type IV alpha subunit blocker
  14. US regulatory status: approved. Mechanism: Dihydrofolate reductase inhibitor.

    Mechanism
    Dihydrofolate reductase inhibitor
  15. US regulatory status: approved. Molecular target: Aromatic-L-amino-acid decarboxylase.

    Target
    Aromatic-L-amino-acid decarboxylase
    Mechanism
    DOPA decarboxylase inhibitor
  16. carfilzomib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: 26S proteasome.

    Target
    26S proteasome
    Mechanism
    26S proteosome inhibitor
  17. US regulatory status: approved. Mechanism: Unknown.

    Mechanism
    Unknown
  18. Development asset linked to Lxo Ireland Designated in public FDA and regional records.

  19. Development asset linked to Lxo Ireland Designated in public FDA and regional records.

  20. Development asset linked to Lxo Ireland Designated in public FDA and regional records.

  21. covid-19 vaccine (inactivated, adjuvanted, adsorbed)

    Antiinfectives for systemic use (J07)

    Antiinfectives for systemic use (J07) compound in Lxo Ireland Designated's portfolio. Mechanism: Biological vaccine - induces immune response.

    Mechanism
    Biological vaccine - induces immune response
  22. dapagliflozin

    Alimentary tract and metabolism (A10)

    US regulatory status: approved. Molecular target: Sodium/glucose cotransporter 2.

    Target
    Sodium/glucose cotransporter 2
    Mechanism
    Sodium/glucose cotransporter 2 inhibitor
  23. US regulatory status: approved. Molecular target: DNA topoisomerase II.

    Target
    DNA topoisomerase II
    Mechanism
    DNA topoisomerase II inhibitor
  24. Development asset linked to Lxo Ireland Designated in public FDA and regional records.

  25. US regulatory status: approved. Molecular target: Voltage-gated calcium channel.

    Target
    Voltage-gated calcium channel
    Mechanism
    Voltage-gated calcium channel modulator
  26. Development asset linked to Lxo Ireland Designated in public FDA and regional records. Molecular target: Insulin receptor.

    Target
    Insulin receptor
    Mechanism
    Insulin receptor agonist
  27. US regulatory status: approved. Molecular target: Enoyl-[acyl-carrier-protein] reductase [NADH] FabI.

    Target
    Enoyl-[acyl-carrier-protein] reductase [NADH] FabI
    Mechanism
    Bacterial enoyl-[acyl-carrier-protein] reductase inhibitor
  28. human heterologous liver cells

    Alimentary tract and metabolism (A16)

    Alimentary tract and metabolism (A16) compound in Lxo Ireland Designated's portfolio.

  29. Development asset linked to Lxo Ireland Designated in public FDA and regional records.

  30. Development asset linked to Lxo Ireland Designated in public FDA and regional records.

  31. Development asset linked to Lxo Ireland Designated in public FDA and regional records. Molecular target: Insulin receptor.

    Target
    Insulin receptor
    Mechanism
    Insulin receptor agonist
  32. Development asset linked to Lxo Ireland Designated in public FDA and regional records.

  33. Development asset linked to Lxo Ireland Designated in public FDA and regional records. Mechanism: Muscarinic acetylcholine receptor M3 antagonist.

    Mechanism
    Muscarinic acetylcholine receptor M3 antagonist
  34. levodopa

    Nervous system (N04)

    US regulatory status: approved. Molecular target: D(3) dopamine receptor.

    Target
    D(3) dopamine receptor
    Mechanism
    Dopamine D3 receptor agonist
  35. Development asset linked to Lxo Ireland Designated in public FDA and regional records.

  36. Development asset linked to Lxo Ireland Designated in public FDA and regional records.

  37. Development asset linked to Lxo Ireland Designated in public FDA and regional records. Mechanism: Mitochondrial complex I (NADH dehydrogenase) inhibitor.

    Mechanism
    Mitochondrial complex I (NADH dehydrogenase) inhibitor
  38. Development asset linked to Lxo Ireland Designated in public FDA and regional records.

  39. paclitaxel

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Tubulin.

    Target
    Tubulin
    Mechanism
    Tubulin inhibitor
  40. US regulatory status: approved. Molecular target: 5-hydroxytryptamine receptor 3A.

    Target
    5-hydroxytryptamine receptor 3A
    Mechanism
    Serotonin 3a (5-HT3a) receptor antagonist
  41. raloxifene

    Genito-urinary system and sex hormones (G03)

    Genito-urinary system and sex hormones (G03) compound in Lxo Ireland Designated's portfolio. Molecular target: Estrogen receptor.

    Target
    Estrogen receptor
    Mechanism
    Estrogen receptor beta modulator
  42. rituximab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: B-lymphocyte antigen CD20.

    Target
    B-lymphocyte antigen CD20
    Mechanism
    B-lymphocyte antigen CD20 binding agent
  43. roflumilast

    Respiratory system (R03)

    US regulatory status: approved. Molecular target: Phosphodiesterase 4.

    Target
    Phosphodiesterase 4
    Mechanism
    Phosphodiesterase 4 inhibitor
  44. rufinamide

    Nervous system (N03)

    US regulatory status: approved. Molecular target: Sodium channel alpha subunit.

    Target
    Sodium channel alpha subunit
    Mechanism
    Sodium channel alpha subunit blocker
  45. Development asset linked to Lxo Ireland Designated in public FDA and regional records.

  46. US regulatory status: approved. Molecular target: Dipeptidyl peptidase 4.

    Target
    Dipeptidyl peptidase 4
    Mechanism
    Dipeptidyl peptidase IV inhibitor
  47. Development asset linked to Lxo Ireland Designated in public FDA and regional records.

  48. Development asset linked to Lxo Ireland Designated in public FDA and regional records.

  49. sufentanil

    Nervous system (N01)

    Nervous system (N01) compound in Lxo Ireland Designated's portfolio. Mechanism: Mu opioid receptor agonist.

    Mechanism
    Mu opioid receptor agonist
  50. Development asset linked to Lxo Ireland Designated in public FDA and regional records.

  51. US regulatory status: approved. Molecular target: DNA topoisomerase 1.

    Target
    DNA topoisomerase 1
    Mechanism
    DNA topoisomerase I, mitochondrial inhibitor
  52. Development asset linked to Lxo Ireland Designated in public FDA and regional records.

  53. ulipristal acetate

    Genito-urinary system and sex hormones (G03)

    US regulatory status: approved. Molecular target: Progesterone receptor.

    Target
    Progesterone receptor
    Mechanism
    Progesterone receptor modulator
  54. Development asset linked to Lxo Ireland Designated in public FDA and regional records.

  55. Development asset linked to Lxo Ireland Designated in public FDA and regional records.