Wednesday, June 10, 2026

Drug profile · INN

methocarbamol

methocarbamol (METHOCARBAMOL) is a carbonic anhydrase i inhibitor. Associated with Regeneron Ireland Designated Activity Company (DAC). Route of administration: injection. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 0
Pipeline programs 1
News articles 0
Drug details — methocarbamol
US status
approved
Class
Route
INJECTION
Patents
0
Programs
1
Data quality
0.89

Quick answer

methocarbamol (METHOCARBAMOL) is a carbonic anhydrase i inhibitor. Associated with Regeneron Ireland Designated Activity Company (DAC). Route of administration: injection. Current US regulatory status: approved.

Key facts

INN methocarbamol
Brand METHOCARBAMOL
Mechanism Carbonic anhydrase I inhibitor
Target Carbonic anhydrase 1
Route INJECTION
Formulation INJECTABLE

Mechanism of action

Carbonic anhydrase I inhibitor

Primary target: Carbonic anhydrase 1

Approval history

Authority Status Date
FDA approved

Pipeline programs

  1. ATM Phase 2 · BRIGHT MINDS BIOSCIENCES · Dual Diagnosis

Related & competitor drugs

  1. acetazolamide Carbonic anhydrase XII inhibitor
  2. acetazolamide sodium Carbonic anhydrase XII inhibitor
  3. dichlorphenamide Carbonic anhydrase XII inhibitor
  4. methazolamide Carbonic anhydrase IV inhibitor
  5. diclofenamide Sensory organs (S01)

Frequently asked questions

What is methocarbamol?

methocarbamol (METHOCARBAMOL) is a carbonic anhydrase i inhibitor. Associated with Regeneron Ireland Designated Activity Company (DAC). Route of administration: injection. Current US regulatory status: approved.

What is the brand name for methocarbamol?

METHOCARBAMOL is a marketed brand name for methocarbamol. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of methocarbamol?

methocarbamol has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.