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Astellas Pharma

Astellas Pharma drug portfolio β€” 52 indexed compounds with therapeutic class and molecular targets from public FDA and regional approval metadata.

2-5-1, Nihonbashi-Honcho, Chuo-Ku, Tokyo 103-8411, JP HQ
12,378 Employees
EMA registrant Type
Company details
Status
Public
HQ
2-5-1, Nihonbashi-Honcho, Chuo-Ku, Tokyo 103-8411, JP
Employees
12,378
Programs
22
Drugs
52
Patents
25
Intelligence Β· Drug Pipeline

Astellas Pharma pipeline

Portfolio lens on 52 drugs and development assets β€” regulatory status, targets, and deep links to NovaPharmaNews drug profiles.

Astellas Pharma drug portfolio β€” 52 indexed compounds with therapeutic class and molecular targets from public FDA and regional approval metadata.

Drug portfolio

52 compounds
  1. abiraterone

    Antineoplastic and immunomodulating agents (L02)

    Antineoplastic and immunomodulating agents (L02) compound in Astellas Pharma's portfolio. Molecular target: Androgen receptor.

    Target
    Androgen receptor
    Mechanism
    Steroid 5-alpha-reductase inhibitor
  2. abiraterone acetate

    Antineoplastic and immunomodulating agents (L02)

    US regulatory status: approved. Molecular target: Steroid 17-alpha-hydroxylase/17,20 lyase.

    Target
    Steroid 17-alpha-hydroxylase/17,20 lyase
    Mechanism
    Cytochrome P450 17A1 inhibitor
  3. apalutamide

    Antineoplastic and immunomodulating agents (L02)

    US regulatory status: approved. Molecular target: Androgen receptor.

    Target
    Androgen receptor
    Mechanism
    Androgen Receptor antagonist
  4. avacincaptad pegol

    Sensory organs (S01)

    Sensory organs (S01) compound in Astellas Pharma's portfolio.

  5. azacitidine

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: DNA (cytosine-5)-methyltransferase 1.

    Target
    DNA (cytosine-5)-methyltransferase 1
    Mechanism
    DNA (cytosine-5)-methyltransferase 3A inhibitor
  6. US regulatory status: approved. Molecular target: Androgen receptor.

    Target
    Androgen receptor
    Mechanism
    Androgen Receptor antagonist
  7. US regulatory status: approved.

  8. capecitabine

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    Thymidylate synthase inhibitor
  9. Development asset linked to Astellas Pharma in public FDA and regional records.

  10. Development asset linked to Astellas Pharma in public FDA and regional records.

  11. US regulatory status: approved. Mechanism: Unknown.

    Mechanism
    Unknown
  12. Development asset linked to Astellas Pharma in public FDA and regional records.

  13. Development asset linked to Astellas Pharma in public FDA and regional records.

  14. docetaxel

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Tubulin.

    Target
    Tubulin
    Mechanism
    Tubulin inhibitor
  15. Development asset linked to Astellas Pharma in public FDA and regional records.

  16. Development asset linked to Astellas Pharma in public FDA and regional records.

  17. enfortumab vedotin

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Astellas Pharma's portfolio. Molecular target: Nectin-4.

    Target
    Nectin-4
    Mechanism
    Tubulin inhibitor
  18. enzalutamide

    Antineoplastic and immunomodulating agents (L02)

    US regulatory status: approved. Molecular target: Androgen receptor.

    Target
    Androgen receptor
    Mechanism
    Androgen Receptor antagonist
  19. US regulatory status: approved. Molecular target: Estrogen receptor.

    Target
    Estrogen receptor
    Mechanism
    Estrogen receptor alpha agonist
  20. fezolinetant

    Genito-urinary system and sex hormones (G02)

    US regulatory status: approved. Molecular target: Neuromedin-K receptor.

    Target
    Neuromedin-K receptor
    Mechanism
    Neurokinin 3 receptor antagonist
  21. filgrastim

    Antineoplastic and immunomodulating agents (L03)

    US regulatory status: approved. Molecular target: Granulocyte colony-stimulating factor receptor.

    Target
    Granulocyte colony-stimulating factor receptor
    Mechanism
    Granulocyte colony stimulating factor receptor agonist
  22. Development asset linked to Astellas Pharma in public FDA and regional records.

  23. US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    Thymidylate synthase inhibitor
  24. Development asset linked to Astellas Pharma in public FDA and regional records.

  25. US regulatory status: approved. Mechanism: DNA polymerase (alpha/delta/epsilon) inhibitor.

    Mechanism
    DNA polymerase (alpha/delta/epsilon) inhibitor
  26. gilteritinib

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Astellas Pharma's portfolio. Molecular target: Receptor-type tyrosine-protein kinase FLT3.

    Target
    Receptor-type tyrosine-protein kinase FLT3
    Mechanism
    Tyrosine-protein kinase receptor FLT3 inhibitor
  27. Development asset linked to Astellas Pharma in public FDA and regional records. Mechanism: Mu opioid receptor agonist.

    Mechanism
    Mu opioid receptor agonist
  28. Development asset linked to Astellas Pharma in public FDA and regional records.

  29. Development asset linked to Astellas Pharma in public FDA and regional records.

  30. Development asset linked to Astellas Pharma in public FDA and regional records.

  31. Development asset linked to Astellas Pharma in public FDA and regional records.

  32. Development asset linked to Astellas Pharma in public FDA and regional records.

  33. mirabegron

    Genito-urinary system and sex hormones (G04)

    US regulatory status: approved. Molecular target: Beta-3 adrenergic receptor.

    Target
    Beta-3 adrenergic receptor
    Mechanism
    Beta-3 adrenergic receptor agonist
  34. nivolumab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Programmed cell death protein 1.

    Target
    Programmed cell death protein 1
    Mechanism
    Programmed cell death protein 1 inhibitor
  35. US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  36. paclitaxel

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Tubulin.

    Target
    Tubulin
    Mechanism
    Tubulin inhibitor
  37. pembrolizumab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Programmed cell death protein 1.

    Target
    Programmed cell death protein 1
    Mechanism
    Programmed cell death protein 1 inhibitor
  38. Development asset linked to Astellas Pharma in public FDA and regional records.

  39. Development asset linked to Astellas Pharma in public FDA and regional records.

  40. US regulatory status: approved. Molecular target: Glucocorticoid receptor.

    Target
    Glucocorticoid receptor
    Mechanism
    Glucocorticoid receptor agonist
  41. US regulatory status: approved. Molecular target: Glucocorticoid receptor.

    Target
    Glucocorticoid receptor
    Mechanism
    Glucocorticoid receptor agonist
  42. Development asset linked to Astellas Pharma in public FDA and regional records.

  43. Development asset linked to Astellas Pharma in public FDA and regional records.

  44. Development asset linked to Astellas Pharma in public FDA and regional records.

  45. Development asset linked to Astellas Pharma in public FDA and regional records.

  46. Development asset linked to Astellas Pharma in public FDA and regional records.

  47. tacrolimus

    Dermatologicals (D11)

    US regulatory status: approved. Molecular target: Peptidyl-prolyl cis-trans isomerase FKBP1A.

    Target
    Peptidyl-prolyl cis-trans isomerase FKBP1A
    Mechanism
    FK506-binding protein 1A inhibitor
  48. Development asset linked to Astellas Pharma in public FDA and regional records.

  49. Development asset linked to Astellas Pharma in public FDA and regional records.

  50. vinflunine

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Astellas Pharma's portfolio. Molecular target: Tubulin.

    Target
    Tubulin
    Mechanism
    Tubulin inhibitor
  51. zolbetuximab

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Astellas Pharma's portfolio. Molecular target: Claudin-18.

    Target
    Claudin-18
    Mechanism
    Claudin-18 binding agent