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Intelligence · Patent portfolio

LEXICON PHARMACEUTICALS Patents

Full USPTO pharma patent portfolio for LEXICON PHARMACEUTICALS — grant dates, expiration, and drug cross-links.

Patents
102
Expiring ≤24m
4

Quick answer

LEXICON PHARMACEUTICALS has 102 pharmaceutical patents in our USPTO PatentsView index (A61K/A61P). 4 expire within 24 months — use filters for patent-cliff planning.

Page 2 of 3

  1. US 7998994

    Solid forms of (1R,2S,3R)-1-(2-(isoxazol-3-yl)-1H-imidazol-4-yl)butane-1,2,3,4-tetraol and methods of their use

    Expires Mon Aug 11 2031 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

  2. US 7968559

    Methods of using 4-phenyl-6-(2,2,2-trifluoro-1-phenylethoxy)pyrimidine-based compounds

    Expires Mon Jun 23 2031 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

  3. US 7968726

    Methods of preparing imidazole-based bicyclic compounds

    Expires Mon Jun 23 2031 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

  4. US 7935796

    Monoclonal antibodies against ANGPTL3

    Expires Mon Apr 28 2031 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

  5. US 7919618

    Synthesis of piperazines, piperidines and related compounds

    Expires Mon Mar 31 2031 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

  6. US 7897763

    Process for the preparation of substituted phenylalanines

    Expires Mon Feb 24 2031 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

  7. US 7875622

    Methods and compositions for treating pulmonary hypertension and related diseases and disorders

    Expires Mon Jan 20 2031 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

  8. US 7855291

    Process for the preparation of substituted phenylalanines

    Expires Mon Dec 16 2030 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

  9. US 7846945

    Piperdine-based inhibitors of sodium glucose co-transporter 2 and methods of their use

    Expires Mon Dec 02 2030 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

  10. US 7825150

    Compositions and methods for treating immunological and inflammatory diseases and disorders

    Expires Mon Oct 28 2030 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

  11. US 7825142

    Heterocyclic compounds, compositions comprising them and methods of their use

    Expires Mon Oct 28 2030 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

  12. US 7812174

    Methods of preparing imidazole-based compounds

    Expires Mon Oct 07 2030 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

  13. US 7781577

    Inhibitors of sodium glucose co-transporter 2 and methods of their use

    Expires Mon Aug 19 2030 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

  14. US 7723345

    Multicyclic amino acid derivatives and methods of their use

    Expires Mon May 20 2030 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

  15. US 7709493

    4-phenyl-6-(2,2,2-trifluoro-1-phenylethoxy)pyrimidine-based compounds and methods of their use

    Expires Mon Apr 29 2030 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

  16. US 7655762

    Monoclonal antibodies against ANGPTL4

    Expires Mon Jan 28 2030 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

  17. US 7649098

    Imidazole-based compounds, compositions comprising them and methods of their use

    Expires Mon Jan 14 2030 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

  18. US 7598280

    Heterocyclic compounds, compositions comprising them and methods of their use

    Expires Mon Oct 01 2029 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

  19. US 7553840

    4-phenyl-6-(2,2,2-trifluoro-1-phenylethoxy)pyrimidine-based compounds and methods of their use

    Expires Mon Jun 25 2029 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

  20. US 7423043

    4-Piperidin-1-yl-7H-pyrrolo[2,3-d]pyrimidine compounds

    Expires Mon Sep 04 2028 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

  21. US 7374932

    Human kinases and polynucleotides encoding the same, and uses thereof

    Expires Mon May 15 2028 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

  22. US 7300949

    Thiazolopyrazoles and methods of their use

    Expires Mon Nov 22 2027 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

  23. US 7268222

    Polynucleotides encoding human transporter proteins

    Expires Mon Sep 06 2027 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

  24. US 7179827

    Thiazoles and methods of their use

    Expires Mon Feb 15 2027 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

  25. US 7057029

    Human ion-exchanger proteins

    Expires Mon Jun 01 2026 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

  26. US 6987178

    Human uncoupling proteins and polynucleotides encoding the same

    Expires Mon Jan 12 2026 00:00:00 GMT+0000 (Coordinated Universal Time)

    expired

  27. US 6929937

    Human transferase proteins and polynucleotides encoding the same

    Expires Mon Aug 11 2025 00:00:00 GMT+0000 (Coordinated Universal Time)

    expired

  28. US 6900045

    Human kinase proteins and polynucleotides encoding the same

    Expires Mon May 26 2025 00:00:00 GMT+0000 (Coordinated Universal Time)

    expired

  29. US 6875587

    Human protease inhibitor and polynucleotides encoding the same

    Expires Mon Mar 31 2025 00:00:00 GMT+0000 (Coordinated Universal Time)

    expired

  30. US 6867291

    Human hemicentin proteins and polynucleotides encoding the same

    Expires Mon Mar 10 2025 00:00:00 GMT+0000 (Coordinated Universal Time)

    expired

  31. US 6864079

    Human kinase and polynucleotides encoding the same

    Expires Mon Mar 03 2025 00:00:00 GMT+0000 (Coordinated Universal Time)

    expired

  32. US 6861241

    Human kinase and polynucleotides encoding the same

    Expires Mon Feb 24 2025 00:00:00 GMT+0000 (Coordinated Universal Time)

    expired

  33. US 6858419

    Human kinases and polynucleotides encoding the same, and uses thereof

    Expires Mon Feb 17 2025 00:00:00 GMT+0000 (Coordinated Universal Time)

    expired

  34. US 6835564

    Human endothelin converting enzyme-like proteins and polynucleotides encoding the same

    Expires Mon Dec 23 2024 00:00:00 GMT+0000 (Coordinated Universal Time)

    expired

  35. US 6815188

    Human kinases and polynucleotides encoding the same

    Expires Mon Nov 04 2024 00:00:00 GMT+0000 (Coordinated Universal Time)

    expired

  36. US 6806073

    Human kinase proteins and polynucleotides encoding the same

    Expires Mon Oct 14 2024 00:00:00 GMT+0000 (Coordinated Universal Time)

    expired

  37. US 6787352

    Polynucleotides encoding human ion-exchanger proteins

    Expires Mon Sep 02 2024 00:00:00 GMT+0000 (Coordinated Universal Time)

    expired

  38. US 6780640

    Human carboxypeptidases and polynucleotides encoding the same

    Expires Mon Aug 19 2024 00:00:00 GMT+0000 (Coordinated Universal Time)

    expired

  39. US 6777221

    Human proteases and polynucleotides encoding the same

    Expires Mon Aug 12 2024 00:00:00 GMT+0000 (Coordinated Universal Time)

    expired

  40. US 6777232

    Human membrane proteins and polynucleotides encoding the same

    Expires Mon Aug 12 2024 00:00:00 GMT+0000 (Coordinated Universal Time)

    expired

  41. US 6767736

    Human ion channel protein and polynucleotides encoding the same

    Expires Mon Jul 22 2024 00:00:00 GMT+0000 (Coordinated Universal Time)

    expired

  42. US 6746861

    Human kinase protein and polynucleotides encoding the same

    Expires Mon Jun 03 2024 00:00:00 GMT+0000 (Coordinated Universal Time)

    expired

  43. US 6602698

    Human kinase proteins and polynucleotides encoding the same

    Expires Mon Jul 31 2023 00:00:00 GMT+0000 (Coordinated Universal Time)

    expired

  44. US 6593125

    Human kinases and polynucleotides encoding the same

    Expires Mon Jul 10 2023 00:00:00 GMT+0000 (Coordinated Universal Time)

    expired

  45. US 6586582

    Human GABA receptor proteins and polynucleotides encoding the same

    Expires Mon Jun 26 2023 00:00:00 GMT+0000 (Coordinated Universal Time)

    expired

  46. US 6583269

    Human protease inhibitor and polynucleotides encoding the same

    Expires Mon Jun 19 2023 00:00:00 GMT+0000 (Coordinated Universal Time)

    expired

  47. US 6555669

    Human transferase proteins and polynucleotides encoding the same

    Expires Mon Apr 24 2023 00:00:00 GMT+0000 (Coordinated Universal Time)

    expired

  48. US 6541252

    Human kinases and polynucleotides encoding the same

    Expires Mon Mar 27 2023 00:00:00 GMT+0000 (Coordinated Universal Time)

    expired

Frequently asked questions

How many patents does LEXICON PHARMACEUTICALS have?

102 published patents match the current filter (all indexed). The full portfolio is indexed from USPTO PatentsView (A61K/A61P).

When do LEXICON PHARMACEUTICALS patents expire?

4 patents in the full portfolio expire within 24 months. Use the expiring filters above or open individual patent pages for grant and expiration dates.

Where does this data come from?

USPTO PatentsView bulk data filtered to pharmaceutical CPC classes (A61K, A61P), cross-linked to NovaPharmaNews company and drug profiles. See our data sources page for methodology.

Data attribution: Data sources · Patent directory

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