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Patents

Browse 41 pharma-relevant patents (US and EP, A61K/A61P) linked to tracked companies. Patent cliff and LOE intelligence for BD teams.

29,054 patents indexed
patent

US 9062007

Cyclic amide BACE-1 inhibitors having a benzamide substituent

Pharmacopeia Drug Discovery, Inc. Β· Granted Tue Jun 23 2015 00:00:00 GMT+0000 (Coordinated Universal Time) Β· Expires Mon Jun 18 2035 00:00:00 GMT+0000 (Coordinated Universal Time)

granted
patent

US 8937093

Heterocyclic aspartyl protease inhibitors

Pharmacopeia Drug Discovery, Inc. Β· Granted Tue Jan 20 2015 00:00:00 GMT+0000 (Coordinated Universal Time) Β· Expires Mon Jan 15 2035 00:00:00 GMT+0000 (Coordinated Universal Time)

granted
patent

US 8778980

Heterocyclic aspartyl protease inhibitors

Pharmacopeia Drug Discovery, Inc. Β· Granted Tue Jul 15 2014 00:00:00 GMT+0000 (Coordinated Universal Time) Β· Expires Mon Jul 10 2034 00:00:00 GMT+0000 (Coordinated Universal Time)

granted
patent

US 8722708

Substituted isoindolines as aspartyl protease inhibitors

Pharmacopeia Drug Discovery, Inc. Β· Granted Tue May 13 2014 00:00:00 GMT+0000 (Coordinated Universal Time) Β· Expires Mon May 08 2034 00:00:00 GMT+0000 (Coordinated Universal Time)

granted
patent

US 8691831

Heterocyclic aspartyl protease inhibitors

Pharmacopeia Drug Discovery, Inc. Β· Granted Tue Apr 08 2014 00:00:00 GMT+0000 (Coordinated Universal Time) Β· Expires Mon Apr 03 2034 00:00:00 GMT+0000 (Coordinated Universal Time)

granted
patent

US 8623867

Cyclic amine BACE-1 inhibitors having a benzamide substituent

Pharmacopeia Drug Discovery, Inc. Β· Granted Tue Jan 07 2014 00:00:00 GMT+0000 (Coordinated Universal Time) Β· Expires Mon Jan 02 2034 00:00:00 GMT+0000 (Coordinated Universal Time)

granted
patent

US 8242112

Heterocyclic aspartyl protease inhibitors

Pharmacopeia Drug Discovery, Inc. Β· Granted Tue Aug 14 2012 00:00:00 GMT+0000 (Coordinated Universal Time) Β· Expires Mon Aug 09 2032 00:00:00 GMT+0000 (Coordinated Universal Time)

granted
patent

US 8207170

Heterocyclic substituted piperazines with CXCR3 antagonist activity

Pharmacopeia Drug Discovery, Inc. Β· Granted Tue Jun 26 2012 00:00:00 GMT+0000 (Coordinated Universal Time) Β· Expires Mon Jun 21 2032 00:00:00 GMT+0000 (Coordinated Universal Time)

granted
patent

US 8178513

Heterocyclic aspartyl protease inhibitors

Pharmacopeia Drug Discovery, Inc. Β· Granted Tue May 15 2012 00:00:00 GMT+0000 (Coordinated Universal Time) Β· Expires Mon May 10 2032 00:00:00 GMT+0000 (Coordinated Universal Time)

granted
patent

US 7985748

ALPHA2C adrenoreceptor agonists

Pharmacopeia Drug Discovery, Inc. Β· Granted Tue Jul 26 2011 00:00:00 GMT+0000 (Coordinated Universal Time) Β· Expires Mon Jul 21 2031 00:00:00 GMT+0000 (Coordinated Universal Time)

granted
patent

US 7964646

3,4-DI-substituted cyclobutene-1,2-diones as CXC-chemokine receptor ligands

Pharmacopeia Drug Discovery, Inc. Β· Granted Tue Jun 21 2011 00:00:00 GMT+0000 (Coordinated Universal Time) Β· Expires Mon Jun 16 2031 00:00:00 GMT+0000 (Coordinated Universal Time)

granted
patent

US 7947720

3,4-di-substituted cyclobutene-1,2-diones as CXC-chemokine receptor ligands

Pharmacopeia Drug Discovery, Inc. Β· Granted Tue May 24 2011 00:00:00 GMT+0000 (Coordinated Universal Time) Β· Expires Mon May 19 2031 00:00:00 GMT+0000 (Coordinated Universal Time)

granted
patent

US 7879838

Heteroaryl substituted pyrazinyl-piperazine-piperidines with CXCR3 antagonist activity

Pharmacopeia Drug Discovery, Inc. Β· Granted Tue Feb 01 2011 00:00:00 GMT+0000 (Coordinated Universal Time) Β· Expires Mon Jan 27 2031 00:00:00 GMT+0000 (Coordinated Universal Time)

granted
patent

US 7868006

Heterocyclic substituted piperazines with CXCR3 antagonist activity

Pharmacopeia Drug Discovery, Inc. Β· Granted Tue Jan 11 2011 00:00:00 GMT+0000 (Coordinated Universal Time) Β· Expires Mon Jan 06 2031 00:00:00 GMT+0000 (Coordinated Universal Time)

granted
patent

US 7799789

Heterocyclic substituted pyridine or phenyl compounds with CXCR3 antagonist activity

Pharmacopeia Drug Discovery, Inc. Β· Granted Tue Sep 21 2010 00:00:00 GMT+0000 (Coordinated Universal Time) Β· Expires Mon Sep 16 2030 00:00:00 GMT+0000 (Coordinated Universal Time)

granted
patent

US 7786149

Thiadiazoles as CXC- and CC- chemokine receptor ligands

Pharmacopeia Drug Discovery, Inc. Β· Granted Tue Aug 31 2010 00:00:00 GMT+0000 (Coordinated Universal Time) Β· Expires Mon Aug 26 2030 00:00:00 GMT+0000 (Coordinated Universal Time)

granted
patent

US 7723340

Haloaryl substituted aminopurines, compositions thereof, and methods of treatment therewit

Pharmacopeia Drug Discovery, Inc. Β· Granted Tue May 25 2010 00:00:00 GMT+0000 (Coordinated Universal Time) Β· Expires Mon May 20 2030 00:00:00 GMT+0000 (Coordinated Universal Time)

granted
patent

US 7566718

Amine-linked pyridyl and phenyl substituted piperazine-piperidines with CXCR3 antagonist a

Pharmacopeia Drug Discovery, Inc. Β· Granted Tue Jul 28 2009 00:00:00 GMT+0000 (Coordinated Universal Time) Β· Expires Mon Jul 23 2029 00:00:00 GMT+0000 (Coordinated Universal Time)

granted
patent

US 7208602

Gamma secretase inhibitors

Pharmacopeia Drug Discovery, Inc. Β· Granted Tue Apr 24 2007 00:00:00 GMT+0000 (Coordinated Universal Time) Β· Expires Mon Apr 19 2027 00:00:00 GMT+0000 (Coordinated Universal Time)

granted
patent

US 7161003

Pyrazolopyrimidines as cyclin dependent kinase inhibitors

Pharmacopeia Drug Discovery, Inc. Β· Granted Tue Jan 09 2007 00:00:00 GMT+0000 (Coordinated Universal Time) Β· Expires Mon Jan 04 2027 00:00:00 GMT+0000 (Coordinated Universal Time)

granted
patent

US 7119200

Pyrazolopyrimidines as cyclin dependent kinase inhibitors

Pharmacopeia Drug Discovery, Inc. Β· Granted Tue Oct 10 2006 00:00:00 GMT+0000 (Coordinated Universal Time) Β· Expires Mon Oct 05 2026 00:00:00 GMT+0000 (Coordinated Universal Time)

granted
patent

US 7084154

2-(aminomethyl) arylamide analgesics

Pharmacopeia Drug Discovery, Inc. Β· Granted Tue Aug 01 2006 00:00:00 GMT+0000 (Coordinated Universal Time) Β· Expires Mon Jul 27 2026 00:00:00 GMT+0000 (Coordinated Universal Time)

granted
patent

US 7084271

Pyrazolopyrimidines as cyclin dependent kinase inhibitors

Pharmacopeia Drug Discovery, Inc. Β· Granted Tue Aug 01 2006 00:00:00 GMT+0000 (Coordinated Universal Time) Β· Expires Mon Jul 27 2026 00:00:00 GMT+0000 (Coordinated Universal Time)

granted
patent

US 7078525

Pyrazolopyrimidines as cyclin dependent kinase inhibitors

Pharmacopeia Drug Discovery, Inc. Β· Granted Tue Jul 18 2006 00:00:00 GMT+0000 (Coordinated Universal Time) Β· Expires Mon Jul 13 2026 00:00:00 GMT+0000 (Coordinated Universal Time)

granted